GPCR Screening

Creative Biogene offers enriched active assay platforms in multiple direct functional readouts, including ligand binding, calcium flux, IP-3/1, cAMP, pERK, GTPγS, reporter assays and internalization assays. GPCR assays in Creative Biogene assist the evaluation of binding and downstream effects of small molecules against a wide variety of GPCR targets. Our GPCR screening assays include over one hundred targets and cover receptors from all major GPCR classes. Whether you're looking for hit identification, selectivity profiling or SAR optimization services, we have all the GPCR drug discovery solutions for you.